2146 |
ENHANCER OF ZESTE 2 POLYCOMB REPRESSIVE COMPLEX 2 SUBUNIT |
EZH2 |
ENX-1 |
ENX1 |
EZH2b |
KMT6 |
KMT6A |
WVS |
WVS2 |
601573 |
3527 |
ENSG00000106462 |
OTTHUMG00000158973 |
2654 |
Q15910 |
NP_004447 |
NM_004456 |
63 |
EZH1 |
Enhancer of zeste homolog 2 |
T25265 |
Histone-lysine N-methyltransferase EZH2 |
BE0009562 |
Initial Gene Query | EZH2 |
Counted Citations from 1950-2000 | 276 |
GuideToPharmacology Gene Category Name | 2.1.1.43 Histone methyltransferases (HMTs) |
GuideToPharmacology Gene Category ID | 871 |
Gene Biotype | PROTEIN_CODING |
NUCLEAR HORMONE RECEPTOR |
CLINICALLY ACTIONABLE |
METHYL TRANSFERASE |
ENZYME |
TRANSCRIPTION FACTOR |
inhibitor (inhibitory) |
Direct Interaction? | True |
Endogenous Drug? | False |
Specific Action of the Ligand | Inhibition |
inhibitor (inhibitory) |
Details of the Assay for Interaction | Inhibition of enzyme function in a biochemical assay using the (activating) Y641N mutant form of EZH2. |
Specific Action of the Ligand | Inhibition |
Endogenous Drug? | False |
EZH2 | Ensembl Gene Name |
Gene Biotype | PROTEIN_CODING |
2146 | Entrez Gene ID |
Initial Gene Query | EZH2 |
Counted Citations from 1950-2000 | 276 |
METHYL TRANSFERASE |
3527 | HUGO Gene ID |
3527 | HUGO Gene Symbol |
enhancer of zeste 2 polycomb repressive complex 2 subunit | HUGO Gene Name |
GuideToPharmacology Gene Category Name | 2.1.1.43 Histone methyltransferases (HMTs) |
GuideToPharmacology Gene Category ID | 871 |
ENZYME |
2146 | CKB Entrez Id |
EZH2 | CKB Gene Synonym |
ENX-1 | CKB Gene Synonym |
2146 | Entrez Gene ID |
63 | CIViC Gene ID |
EZH2 | DrugBank Gene Name |
Q15910 | UniProt Accession |
2146 | Entrez Gene Id |
2146 | OncoKB Entrez Id |
ENX-1 | OncoKB Gene Synonym |
ENX1 | OncoKB Gene Synonym |
ENSG00000106462 | Ensembl Gene ID |
ENX-1 | Human Protein Atlas Gene Synonym |
EZH1 | Human Protein Atlas Gene Synonym |
ENZYME |
Histone-lysine N-methyltransferase EZH2 | Gene Name |
Q15910 | UniProt ID |
NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR |
EZH2 | Gene Symbol |
CLINICALLY ACTIONABLE |
EZH2 | TTD Gene Abbreviation |
T25265 | TTD Target ID |
CLINICALLY ACTIONABLE |
CLINICALLY ACTIONABLE |
CLINICALLY ACTIONABLE |
CLINICALLY ACTIONABLE |