780 |
DISCOIDIN DOMAIN RECEPTOR TYROSINE KINASE 1 |
DDR1 |
CAK |
CD167 |
DDR |
EDDR1 |
HGK2 |
MCK10 |
NEP |
NTRK4 |
PTK3 |
PTK3A |
RTK6 |
TRKE |
600408 |
2730 |
ENSG00000204580 |
OTTHUMG00000031236 |
Q08345 |
EPITHELIAL DISCOIDIN DOMAIN-CONTAINING RECEPTOR 1 |
DDR1_HUMAN |
ENSG00000137332 |
ENSG00000215522 |
ENSG00000234078 |
ENSG00000230456 |
1843 |
NM_001202521 |
NP_001945 |
ENSG00000137332; ENSG00000204580; ENSG00000215522; ENSG00000230456; ENSG00000234078 |
BE0001124 |
EPITHELIAL DISCOIDIN DOMAIN RECEPTOR 1 PRECURSOR (EC 2.7.1.112) (TYROSINE KINASE DDR) (DISCOIDIN RECEPTOR TYROSINE KINASE) (TYROSINE- PROTEIN KINASE CAK) (CELL ADHESION KINASE) (TRK E) (PROTEIN-TYROSINE KINASE RTK 6) (CD167A ANTIGEN) (HGK2). [SOURCE:UNIPR |
Epithelial discoidin domain receptor 1 |
T09185 |
Uniprot Evidence | 1: Evidence at protein level |
Human Readable Name | DRUGGABLE GENOME |
Interpro Name | Serine-threonine/tyrosine-protein kinase catalytic domain |
Interpro Acc | IPR001245 |
Interpro Type | Domain |
Human Readable Name | KINASE |
Uniprot Status | Swiss-Prot |
Interpro Short Name | Ser-Thr/Tyr_kinase_cat_dom |
Target Class | Receptors |
Target Subclass | EC:2.7.10.1 |
GuideToPharmacology Gene Category Name | Type XVI RTKs: DDR (collagen receptor) family |
GuideToPharmacology Gene Category ID | 331 |
Target Subclass | Kinase |
Transmembrane Helix Count | 1 |
Target Main Class | Receptors |
Gene Biotype | PROTEIN_CODING |
KINASE |
TYROSINE KINASE |
DRUGGABLE GENOME |
CLINICALLY ACTIONABLE |
antagonist (inhibitory) |
inhibitor (inhibitory) |
Specific Action of the Ligand | Inhibition |
Endogenous Drug? | False |
Direct Interaction? | False |
inhibitor (inhibitory) |
Details of the Assay for Interaction | Binding constant determined by KINOMEScan assay. |
Specific Action of the Ligand | Inhibition |
Endogenous Drug? | False |
inhibitor (inhibitory) |
Specific Action of the Ligand | Inhibition |
Endogenous Drug? | False |
Direct Interaction? | False |
DDR1 | Ensembl Gene Name |
Gene Biotype | PROTEIN_CODING |
DDR1_HUMAN | Uniprot Id |
EPITHELIAL DISCOIDIN DOMAIN-CONTAINING RECEPTOR 1 | Uniprot Protein Name |
780 | Entrez Gene Id |
Uniprot Evidence | 1: Evidence at protein level |
Human Readable Name | DRUGGABLE GENOME |
Interpro Name | Serine-threonine/tyrosine-protein kinase catalytic domain |
KINASE, DRUGGABLE GENOME |
DDR1 | Gene Symbol |
Target Class | Receptors |
Target Subclass | EC:2.7.10.1 |
ENSG00000137332 | Ensembl Gene Id |
EPITHELIAL DISCOIDIN DOMAIN RECEPTOR 1 PRECURSOR (EC 2.7.1.112) (TYROSINE KINASE DDR) (DISCOIDIN RECEPTOR TYROSINE KINASE) (TYROSINE- PROTEIN KINASE CAK) (CELL ADHESION KINASE) (TRK E) (PROTEIN-TYROSINE KINASE RTK 6) (CD167A ANTIGEN) (HGK2). [SOURCE:UNIPR | Description |
DDR1 | Display Id |
Human Readable Name | DRUGGABLE GENOME |
DRUGGABLE GENOME |
ENSG00000137332; ENSG00000204580; ENSG00000215522; ENSG00000230456; ENSG00000234078 | Ensembl Gene Id |
Q08345 | Uniprot Accession |
DDR1_HUMAN | Uniprot Id |
Target Subclass | Kinase |
Transmembrane Helix Count | 1 |
Target Main Class | Receptors |
2730 | HUGO Gene ID |
2730 | HUGO Gene Symbol |
discoidin domain receptor tyrosine kinase 1 | HUGO Gene Name |
GuideToPharmacology Gene Category Name | Type XVI RTKs: DDR (collagen receptor) family |
GuideToPharmacology Gene Category ID | 331 |
DDR1 | DrugBank Gene Name |
Q08345 | UniProt Accession |
780 | Entrez Gene Id |
ENSG00000204580 | Gene Symbol |
DDR1 | Ensembl Id |
DRUGGABLE GENOME |
Epithelial discoidin domain-containing receptor 1 | Gene Name |
Q08345 | UniProt ID |
KINASE |
780 | Gene ID |
CAK | dGene Synonym |
CD167 | dGene Synonym |
KINASE, TYROSINE KINASE |
DDR1 | TTD Gene Abbreviation |
T09185 | TTD Target ID |
CLINICALLY ACTIONABLE |