1131 |
CHOLINERGIC RECEPTOR MUSCARINIC 3 |
CHRM3 |
EGBRS |
HM3 |
PBS |
118494 |
1952 |
ENSG00000133019 |
OTTHUMG00000039649 |
P20309 |
MUSCARINIC ACETYLCHOLINE RECEPTOR M3 |
ACM3_HUMAN |
MUSCARINIC ACETYLCHOLINE RECEPTOR M3. [SOURCE:UNIPROT/SWISSPROT;ACC:P20309] |
T67684 |
Uniprot Status | Swiss-Prot |
Interpro Acc | IPR000276 |
Interpro Type | Family |
Interpro Name | GPCR, rhodopsin-like, 7TM |
Uniprot Evidence | 1: Evidence at protein level |
Human Readable Name | DRUGGABLE GENOME |
Interpro Short Name | 7TM_GPCR_Rhodpsn |
Human Readable Name | G PROTEIN COUPLED RECEPTOR |
Transmembrane Helix Count | 7 |
Target Subclass | GPCR |
Target Subclass | Rhodopsin |
Target Main Class | Receptors |
Target Class | Receptors |
Gene Biotype | PROTEIN_CODING |
G PROTEIN COUPLED RECEPTOR |
DRUGGABLE GENOME |
antagonist (inhibitory) |
Mechanism of Interaction | Muscarinic acetylcholine receptor M3 antagonist |
Direct Interaction | yes |
antagonist (inhibitory) |
Mechanism of Interaction | Muscarinic acetylcholine receptor M3 antagonist |
Direct Interaction | yes |
Trial Name | SVT-40776 |
antagonist (inhibitory) |
Mechanism of Interaction | Muscarinic acetylcholine receptor M3 antagonist |
Direct Interaction | yes |
Trial Name | transdermal oxybutynin patch, oxybutynin topical gel,Oxytrol, Kentera, Gelnique |
antagonist (inhibitory) |
Mechanism of Interaction | Muscarinic acetylcholine receptor M3 antagonist |
Direct Interaction | yes |
antagonist (inhibitory) |
Direct Interaction | yes |
Mechanism of Interaction | Muscarinic acetylcholine receptor M3 antagonist |
antagonist (inhibitory) |
Mechanism of Interaction | Muscarinic acetylcholine receptor M3 antagonist |
Direct Interaction | yes |
antagonist (inhibitory) |
Mechanism of Interaction | Muscarinic acetylcholine receptor M3 antagonist |
Direct Interaction | yes |
antagonist (inhibitory) |
Direct Interaction | yes |
Mechanism of Interaction | Muscarinic acetylcholine receptor M3 antagonist |
antagonist (inhibitory) |
Mechanism of Interaction | Muscarinic acetylcholine receptor M3 antagonist |
Direct Interaction | yes |
antagonist (inhibitory) |
Mechanism of Interaction | Muscarinic acetylcholine receptor M3 antagonist |
Direct Interaction | yes |
antagonist (inhibitory) |
Novel drug target | Established target |
Trial Name | - |
antagonist (inhibitory) |
Mechanism of Interaction | Muscarinic acetylcholine receptor M3 antagonist |
Direct Interaction | yes |
antagonist (inhibitory) |
Trial Name | fesoterodine fumarate, SPM 907,Toviaz |
Novel drug target | Established target |
antagonist (inhibitory) |
Trial Name | - |
Novel drug target | Established target |
antagonist (inhibitory) |
Novel drug target | Established target |
Trial Name | - |
antagonist (inhibitory) |
Mechanism of Interaction | Muscarinic acetylcholine receptor M3 antagonist |
Direct Interaction | yes |
Trial Name | inhaled atropine |
antagonist (inhibitory) |
Mechanism of Interaction | Muscarinic acetylcholine receptor M3 antagonist |
Direct Interaction | yes |
antagonist (inhibitory) |
Mechanism of Interaction | Muscarinic acetylcholine receptor M3 antagonist |
Direct Interaction | yes |
antagonist (inhibitory) |
Mechanism of Interaction | Muscarinic acetylcholine receptor M3 antagonist |
Direct Interaction | yes |
antagonist (inhibitory) |
Mechanism of Interaction | Muscarinic acetylcholine receptor M3 antagonist |
Direct Interaction | yes |
antagonist (inhibitory) |
Mechanism of Interaction | Muscarinic acetylcholine receptor M3 antagonist |
Direct Interaction | yes |
antagonist (inhibitory) |
Direct Interaction | yes |
Mechanism of Interaction | Muscarinic acetylcholine receptor M3 antagonist |
antagonist (inhibitory) |
Mechanism of Interaction | Muscarinic acetylcholine receptor M3 antagonist |
Direct Interaction | yes |
antagonist (inhibitory) |
Direct Interaction | yes |
Mechanism of Interaction | Muscarinic acetylcholine receptor M3 antagonist |
agonist (activating) |
Mechanism of Interaction | Muscarinic acetylcholine receptor M3 agonist |
Direct Interaction | yes |
agonist (activating) |
Direct Interaction | yes |
Mechanism of Interaction | Muscarinic acetylcholine receptor M3 agonist |
antagonist (inhibitory) |
Mechanism of Interaction | Muscarinic acetylcholine receptor M3 antagonist |
Direct Interaction | yes |
antagonist (inhibitory) |
Mechanism of Interaction | Muscarinic acetylcholine receptor M3 antagonist |
Direct Interaction | yes |
antagonist (inhibitory) |
Mechanism of Interaction | Muscarinic acetylcholine receptor M3 antagonist |
Direct Interaction | yes |
antagonist (inhibitory) |
Mechanism of Interaction | Muscarinic acetylcholine receptor M3 antagonist |
Direct Interaction | yes |
agonist (activating) |
Mechanism of Interaction | Muscarinic acetylcholine receptor M3 agonist |
Direct Interaction | yes |
antagonist (inhibitory) |
Mechanism of Interaction | Muscarinic acetylcholine receptor M3 antagonist |
Direct Interaction | yes |
antagonist (inhibitory) |
Mechanism of Interaction | Muscarinic acetylcholine receptor M3 antagonist |
Direct Interaction | yes |
antagonist (inhibitory) |
Mechanism of Interaction | Muscarinic acetylcholine receptor M3 antagonist |
Direct Interaction | yes |
antagonist (inhibitory) |
Mechanism of Interaction | Muscarinic acetylcholine receptor M3 antagonist |
Direct Interaction | yes |
antagonist (inhibitory) |
Mechanism of Interaction | Muscarinic acetylcholine receptor M3 antagonist |
Direct Interaction | yes |
antagonist (inhibitory) |
Direct Interaction | yes |
Mechanism of Interaction | Muscarinic acetylcholine receptor M3 antagonist |
agonist (activating) |
Direct Interaction | yes |
Mechanism of Interaction | Muscarinic acetylcholine receptor M3 agonist |
agonist (activating) |
Mechanism of Interaction | Muscarinic acetylcholine receptor M3 agonist |
Direct Interaction | yes |
agonist (activating) |
Novel drug target | Established target |
Trial Name | THVD-201 |
Mechanism of Interaction | Muscarinic acetylcholine receptor M3 agonist |
antagonist (inhibitory) |
Novel drug target | Established target |
Trial Name | - |
antagonist (inhibitory) |
Novel drug target | Established target |
Trial Name | - |
antagonist (inhibitory) |
Direct Interaction | yes |
Mechanism of Interaction | Muscarinic acetylcholine receptor M3 antagonist |
antagonist (inhibitory) |
Trial Name | - |
Novel drug target | Established target |
antagonist (inhibitory) |
Trial Name | Silenor (SO-101) |
Novel drug target | Established target |
agonist (activating) |
Mechanism of Interaction | Muscarinic acetylcholine receptor M3 agonist |
Direct Interaction | yes |
antagonist (inhibitory) |
Mechanism of Interaction | Muscarinic acetylcholine receptor M3 antagonist |
Direct Interaction | yes |
antagonist (inhibitory) |
Trial Name | - |
Novel drug target | Established target |
antagonist (inhibitory) |
Mechanism of Interaction | Muscarinic acetylcholine receptor antagonist |
Direct Interaction | yes |
antagonist (inhibitory) |
Trial Name | Aclidinium |
Novel drug target | Established target |
n/a |
Novel drug target | Established target |
Trial Name | - |
antagonist (inhibitory) |
Mechanism of Interaction | Muscarinic acetylcholine receptor antagonist |
Direct Interaction | yes |
antagonist (inhibitory) |
Direct Interaction | yes |
Mechanism of Interaction | Muscarinic acetylcholine receptor M3 antagonist |
antagonist (inhibitory) |
Trial Name | olanzapine,Zyprexa, Zypadhera, Zyprexa Relprevv |
Novel drug target | Established target |
Trial Name | Olanzapine/fluoxetine combination,Symbyax (Zyprexa/Prozac) |
CHRM3 | Ensembl Gene Name |
Gene Biotype | PROTEIN_CODING |
1131 | Entrez Gene Id |
P20309 | Uniprot Accession |
ACM3_HUMAN | Uniprot Id |
Uniprot Status | Swiss-Prot |
Interpro Acc | IPR000276 |
Interpro Type | Family |
G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME |
1131 | Entrez Gene Id |
P20309 | Uniprot Accession |
ACM3_HUMAN | Uniprot Id |
Transmembrane Helix Count | 7 |
Target Subclass | GPCR |
Target Subclass | Rhodopsin |
CHRM3 | Gene Symbol |
Target Class | Receptors |
Target Subclass | GPCR |
Target Subclass | Rhodopsin |
CHRM3 | Display Id |
ENSG00000133019 | Ensembl Gene Id |
MUSCARINIC ACETYLCHOLINE RECEPTOR M3. [SOURCE:UNIPROT/SWISSPROT;ACC:P20309] | Description |
Human Readable Name | DRUGGABLE GENOME |
DRUGGABLE GENOME |
CHRM3 | GENE_SYMBOL |
Muscarinic acetylcholine receptor M3 | UNIPROT |
ENSG00000133019 | Gene Symbol |
CHRM3 | Ensembl Id |
DRUGGABLE GENOME |
1131 | Gene ID |
EGBRS | dGene Synonym |
HM3 | dGene Synonym |
G PROTEIN COUPLED RECEPTOR |
CHRM3 | TTD Gene Abbreviation |
T67684 | TTD Target ID |