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BRD2 Gene Record

  • Summary
  • Interactions
  • Claims
  • BRD2 6046 Druggable Genome

    Alternate Names:

    6046
    BROMODOMAIN CONTAINING 2
    BRD2
    BRD2-IT1
    D6S113E
    FSH
    FSRG1
    NAT
    O27.1.1
    RING3
    RNF3
    601540
    1103
    ENSG00000204256
    OTTHUMG00000031241
    Bromodomain-containing protein 2
    T86399
    KIAA9001

    Gene Info:

    Gene Biotype PROTEIN_CODING
    (3 More Sources)

    Gene Categories: Category Details

    KINASE
    SERINE THREONINE KINASE
    DRUGGABLE GENOME

    Publications:

    Filippakopoulos et al., 2012, Benzodiazepines and benzotriazepines as protein interaction inhibitors targeting bromodomains of the BET family., Bioorg. Med. Chem.
    Chung CW et al., 2012, Fragment-based discovery of bromodomain inhibitors part 1: inhibitor binding modes and implications for lead discovery., J Med Chem
  • CHEMBL52030   BRD2

    Interaction Score: 5.89

    Interaction Types & Directionality:
    n/a

    Interaction Info:

    PMIDs:
    22137933


    Sources:
    DTC

  • ABBV-744   BRD2

    Interaction Score: 2.94

    Interaction Types & Directionality:
    n/a

    Interaction Info:

    PMIDs:
    None found


    Sources:
    TTD

  • BIRABRESIB   BRD2

    Interaction Score: 2.21

    Interaction Types & Directionality:
    n/a

    Interaction Info:

    PMIDs:
    None found


    Sources:
    TTD

  • ALPRAZOLAM   BRD2

    Interaction Score: 0.59

    Interaction Types & Directionality:
    n/a

    Interaction Info:

    PMIDs:
    22137933


    Sources:
    DTC

  • TRIAZOLAM   BRD2

    Interaction Score: 0.59

    Interaction Types & Directionality:
    n/a

    Interaction Info:

    PMIDs:
    22137933


    Sources:
    DTC

  • MIDAZOLAM   BRD2

    Interaction Score: 0.48

    Interaction Types & Directionality:
    n/a

    Interaction Info:

    PMIDs:
    22137933


    Sources:
    DTC

  • ACETAMINOPHEN   BRD2

    Interaction Score: 0.45

    Interaction Types & Directionality:
    n/a

    Interaction Info:

    PMIDs:
    22136404


    Sources:
    DTC

  • Ensembl: ENSG00000204256

    • Version: 101_38

    Alternate Names:
    BRD2 Ensembl Gene Name

    Gene Info:
    Gene Biotype PROTEIN_CODING

    Publications:

  • NCI: BRD2

    • Version: 14-September-2017

    Alternate Names:

    Gene Info:

    Publications:
    Ostrowski et al., 1998, Stimulation of p85/RING3 kinase in multiple organs after systemic administration of mitogens into mice., Oncogene

  • DTC: BRD2

    • Version: 02-September-2020

    Alternate Names:

    Gene Info:

    Publications:
    Filippakopoulos et al., 2012, Benzodiazepines and benzotriazepines as protein interaction inhibitors targeting bromodomains of the BET family., Bioorg. Med. Chem.
    Chung CW et al., 2012, Fragment-based discovery of bromodomain inhibitors part 1: inhibitor binding modes and implications for lead discovery., J Med Chem

  • HingoraniCasas: ENSG00000204256

    • Version: 31-May-2017

    Alternate Names:
    ENSG00000204256 Gene Symbol
    BRD2 Ensembl Id

    Gene Info:

    Gene Categories:
    DRUGGABLE GENOME

    Publications:

  • GO: BRD2

    • Version: 01-February-2022

    Alternate Names:
    KIAA9001 GO Gene Synonym
    RING3 GO Gene Synonym

    Gene Info:

    Gene Categories:
    SERINE THREONINE KINASE

    Publications:

  • dGene: BRD2

    • Version: 27-Jun-2013

    Alternate Names:
    6046 Gene ID
    D6S113E dGene Synonym
    FSH dGene Synonym

    Gene Info:

    Gene Categories:
    KINASE, SERINE THREONINE KINASE

    Publications:

  • TTD: Bromodomain-containing protein 2

    • Version: 2020.06.01

    Alternate Names:
    BRD2 TTD Gene Abbreviation
    T86399 TTD Target ID

    Gene Info:

    Publications:

Disclaimer: This resource is intended for purely research purposes. It should not be used for emergencies or medical or professional advice.

A finding of a drug-gene interaction or potentially druggable category does not necessarily indicate effectiveness (or lack thereof) of any drug or treatment regimen. A finding of no interaction or no potentially druggable category does not necessarily indicate lack of effectiveness of any drug or treatment regimen. Drug-gene interactions or potentially druggable categories are not presented in ranked order of potential or predicted efficacy.

The dgidb.org website does not provide any medical or healthcare products, services or advice, and is not for medical emergencies or urgent situations. IF YOU THINK YOU MAY HAVE A MEDICAL EMERGENCY, CALL YOUR DOCTOR OR 911 IMMEDIATELY. Information contained on this website is not a substitute for a doctor's medical judgment or advice. We recommend that you discuss your specific, individual health concerns with your doctor or health care professional.

DGIdb (v4.2.0 - sha1 afd9f30b) • Last updated 2020-10-21