DGIdb - BRD2 Gene Record

BRD2 6046 Druggable Genome

Alternate Names:

6046
BROMODOMAIN CONTAINING 2
BRD2
BRD2-IT1
D6S113E
FSH
FSRG1
NAT
O27.1.1
RING3
RNF3
601540
1103
ENSG00000204256
OTTHUMG00000031241
Bromodomain-containing protein 2
T86399
KIAA9001

Gene Info:

Gene Biotype	PROTEIN_CODING

(3 More Sources)

Gene Categories: Category Details

KINASE
SERINE THREONINE KINASE
DRUGGABLE GENOME

Publications:

Filippakopoulos et al., 2012, Benzodiazepines and benzotriazepines as protein interaction inhibitors targeting bromodomains of the BET family., Bioorg. Med. Chem.
Chung CW et al., 2012, Fragment-based discovery of bromodomain inhibitors part 1: inhibitor binding modes and implications for lead discovery., J Med Chem

CHEMBL52030 BRD2

Interaction Score: 5.89

Interaction Types & Directionality:

n/a

Interaction Info:

PMIDs:
22137933

Sources:
DTC
ABBV-744 BRD2

Interaction Score: 2.94

Interaction Types & Directionality:

n/a

Interaction Info:

PMIDs:
None found

Sources:
TTD
BIRABRESIB BRD2

Interaction Score: 2.21

Interaction Types & Directionality:

n/a

Interaction Info:

PMIDs:
None found

Sources:
TTD
ALPRAZOLAM BRD2

Interaction Score: 0.59

Interaction Types & Directionality:

n/a

Interaction Info:

PMIDs:
22137933

Sources:
DTC
TRIAZOLAM BRD2

Interaction Score: 0.59

Interaction Types & Directionality:

n/a

Interaction Info:

PMIDs:
22137933

Sources:
DTC
MIDAZOLAM BRD2

Interaction Score: 0.48

Interaction Types & Directionality:

n/a

Interaction Info:

PMIDs:
22137933

Sources:
DTC
ACETAMINOPHEN BRD2

Interaction Score: 0.45

Interaction Types & Directionality:

n/a

Interaction Info:

PMIDs:
22136404

Sources:
DTC

Ensembl: ENSG00000204256
- Version: 101_38
Alternate Names:

BRD2 Ensembl Gene Name

Gene Info:

Gene Biotype PROTEIN_CODING

Publications:
NCI: BRD2
- Version: 14-September-2017
Alternate Names:

Gene Info:

Publications:

Ostrowski et al., 1998, Stimulation of p85/RING3 kinase in multiple organs after systemic administration of mitogens into mice., Oncogene

DTC: BRD2

Version: 02-September-2020

Alternate Names:

Gene Info:

Publications:

Filippakopoulos et al., 2012, Benzodiazepines and benzotriazepines as protein interaction inhibitors targeting bromodomains of the BET family., Bioorg. Med. Chem.

Chung CW et al., 2012, Fragment-based discovery of bromodomain inhibitors part 1: inhibitor binding modes and implications for lead discovery., J Med Chem

HingoraniCasas: ENSG00000204256
- Version: 31-May-2017
Alternate Names:

ENSG00000204256 Gene Symbol

BRD2 Ensembl Id

Gene Info:

Gene Categories:

DRUGGABLE GENOME

Publications:
GO: BRD2
- Version: 01-February-2022
Alternate Names:

KIAA9001 GO Gene Synonym

RING3 GO Gene Synonym

Gene Info:

Gene Categories:

SERINE THREONINE KINASE

Publications:
dGene: BRD2
- Version: 27-Jun-2013
Alternate Names:

6046 Gene ID

D6S113E dGene Synonym

FSH dGene Synonym

Gene Info:

Gene Categories:

KINASE, SERINE THREONINE KINASE

Publications:
TTD: Bromodomain-containing protein 2
- Version: 2020.06.01
Alternate Names:

BRD2 TTD Gene Abbreviation

T86399 TTD Target ID

Gene Info:

Publications:

6046	Gene ID
D6S113E	dGene Synonym
FSH	dGene Synonym

BRD2	TTD Gene Abbreviation
T86399	TTD Target ID

BRD2 Gene Record

BRD2 6046 Druggable Genome

Alternate Names:

Gene Info:

Gene Categories: Category Details

Publications:

CHEMBL52030 BRD2

Interaction Types & Directionality: n/a

Interaction Info:

PMIDs: 22137933

Sources: DTC

ABBV-744 BRD2

Interaction Types & Directionality: n/a

Interaction Info:

PMIDs: None found

Sources: TTD

BIRABRESIB BRD2

Interaction Types & Directionality: n/a

Interaction Info:

PMIDs: None found

Sources: TTD

ALPRAZOLAM BRD2

Interaction Types & Directionality: n/a

Interaction Info:

PMIDs: 22137933

Sources: DTC

TRIAZOLAM BRD2

Interaction Types & Directionality: n/a

Interaction Info:

PMIDs: 22137933

Sources: DTC

MIDAZOLAM BRD2

Interaction Types & Directionality: n/a

Interaction Info:

PMIDs: 22137933

Sources: DTC

ACETAMINOPHEN BRD2

Interaction Types & Directionality: n/a

Interaction Info:

PMIDs: 22136404

Sources: DTC

Ensembl: ENSG00000204256

Alternate Names: BRD2 Ensembl Gene Name

Gene Info: Gene Biotype PROTEIN_CODING

Publications:

NCI: BRD2

Alternate Names:

Gene Info:

Publications: Ostrowski et al., 1998, Stimulation of p85/RING3 kinase in multiple organs after systemic administration of mitogens into mice., Oncogene

DTC: BRD2

Alternate Names:

Gene Info:

HingoraniCasas: ENSG00000204256

Alternate Names: ENSG00000204256 Gene Symbol BRD2 Ensembl Id

Gene Info:

Gene Categories: DRUGGABLE GENOME

Publications:

GO: BRD2

Alternate Names: KIAA9001 GO Gene Synonym RING3 GO Gene Synonym

Gene Info:

Gene Categories: SERINE THREONINE KINASE

Publications:

dGene: BRD2

Alternate Names: 6046 Gene ID D6S113E dGene Synonym FSH dGene Synonym

Gene Info:

Gene Categories: KINASE, SERINE THREONINE KINASE

Publications:

TTD: Bromodomain-containing protein 2

Alternate Names: BRD2 TTD Gene Abbreviation T86399 TTD Target ID

Gene Info:

Publications:

Interaction Types & Directionality:

n/a

PMIDs:
22137933

Sources:
DTC

Interaction Types & Directionality:

n/a

PMIDs:
None found

Sources:
TTD

Interaction Types & Directionality:

n/a

PMIDs:
None found

Sources:
TTD

Interaction Types & Directionality:

n/a

PMIDs:
22137933

Sources:
DTC

Interaction Types & Directionality:

n/a

PMIDs:
22137933

Sources:
DTC

Interaction Types & Directionality:

n/a

PMIDs:
22137933

Sources:
DTC

Interaction Types & Directionality:

n/a

PMIDs:
22136404

Sources:
DTC

Alternate Names:

BRD2 Ensembl Gene Name

Gene Info:

Gene Biotype PROTEIN_CODING

Publications:

Ostrowski et al., 1998, Stimulation of p85/RING3 kinase in multiple organs after systemic administration of mitogens into mice., Oncogene

Alternate Names:

ENSG00000204256 Gene Symbol

BRD2 Ensembl Id

Gene Categories:

DRUGGABLE GENOME

Alternate Names:

KIAA9001 GO Gene Synonym

RING3 GO Gene Synonym

Gene Categories:

SERINE THREONINE KINASE

Alternate Names:

6046 Gene ID

D6S113E dGene Synonym

FSH dGene Synonym

Gene Categories:

KINASE, SERINE THREONINE KINASE

Alternate Names:

BRD2 TTD Gene Abbreviation

T86399 TTD Target ID