552 |
ARGININE VASOPRESSIN RECEPTOR 1A |
AVPR1A |
AVPR V1a |
AVPR1 |
V1aR |
600821 |
895 |
ENSG00000166148 |
OTTHUMG00000169980 |
P37288 |
V1AR_HUMAN |
VASOPRESSIN V1A RECEPTOR (V1AR) (VASCULAR/HEPATIC-TYPE ARGININE VASOPRESSIN RECEPTOR) (ANTIDIURETIC HORMONE RECEPTOR 1A) (AVPR V1A). [SOURCE:UNIPROT/SWISSPROT;ACC:P37288] |
ANTIDIURETIC HORMONE RECEPTOR 1A |
VASOPRESSIN V1A RECEPTOR |
VASCULAR/HEPATIC-TYPE ARGININE VASOPRESSIN RECEPTOR |
T79232 |
Target Class | Receptors |
Target Subclass | GPCR |
Target Subclass | Rhodopsin |
Human Readable Name | DRUGGABLE GENOME |
Transmembrane Helix Count | 7 |
Target Main Class | Receptors |
Human Readable Name | G PROTEIN COUPLED RECEPTOR |
Uniprot Evidence | 1: Evidence at protein level |
Uniprot Status | Swiss-Prot |
Interpro Name | GPCR, rhodopsin-like, 7TM |
Interpro Type | Family |
Interpro Acc | IPR000276 |
Interpro Short Name | 7TM_GPCR_Rhodpsn |
Gene Biotype | PROTEIN_CODING |
CELL SURFACE |
G PROTEIN COUPLED RECEPTOR |
DRUGGABLE GENOME |
antagonist (inhibitory) |
Mechanism of Interaction | Vasopressin V1a receptor antagonist |
Direct Interaction | yes |
agonist (activating) |
Mechanism of Interaction | Vasopressin V1a receptor agonist |
Direct Interaction | yes |
antagonist (inhibitory) |
Mechanism of Interaction | Vasopressin V1a receptor antagonist |
Direct Interaction | yes |
antagonist (inhibitory) |
Direct Interaction | yes |
Mechanism of Interaction | Vasopressin V1a receptor antagonist |
antagonist (inhibitory) |
Mechanism of Interaction | Vasopressin V1a receptor antagonist |
Direct Interaction | yes |
agonist (activating) |
Novel drug target | Established target |
Trial Name | - |
Mechanism of Interaction | Vasopressin receptor agonist |
antagonist (inhibitory) |
agonist (activating) |
Mechanism of Interaction | Vasopressin V1a receptor agonist |
Direct Interaction | yes |
agonist (activating) |
Direct Interaction | yes |
Mechanism of Interaction | Vasopressin receptor agonist |
agonist (activating) |
AVPR1A | Ensembl Gene Name |
Gene Biotype | PROTEIN_CODING |
VASOPRESSIN V1A RECEPTOR (V1AR) (VASCULAR/HEPATIC-TYPE ARGININE VASOPRESSIN RECEPTOR) (ANTIDIURETIC HORMONE RECEPTOR 1A) (AVPR V1A). [SOURCE:UNIPROT/SWISSPROT;ACC:P37288] | Description |
AVPR1A | Display Id |
ENSG00000166148 | Ensembl Gene Id |
Human Readable Name | DRUGGABLE GENOME |
DRUGGABLE GENOME |
AVPR1A | Gene Symbol |
Target Class | Receptors |
Target Subclass | GPCR |
Target Subclass | Rhodopsin |
AVPR1A | Gene Symbol |
552 | Entrez Gene Id |
ENSG00000166148 | Ensembl Gene Id |
Target Subclass | GPCR |
Transmembrane Helix Count | 7 |
Target Subclass | Rhodopsin |
AVPR1A | Uniprot Gene Name |
P37288 | Uniprot Accession |
552 | Entrez Gene Id |
Uniprot Evidence | 1: Evidence at protein level |
Human Readable Name | DRUGGABLE GENOME |
Human Readable Name | G PROTEIN COUPLED RECEPTOR |
G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME |
V1AR | TTD Gene Abbreviation |
T79232 | TTD Target ID |
AVPR1 | GENE_SYMBOL |
AVPR1A | GENE_SYMBOL |
Vasopressin V1a receptor | UNIPROT |
ENSG00000166148 | Gene Symbol |
AVPR1A | Ensembl Id |
DRUGGABLE GENOME |
AVPR1 | GO Gene Synonym |
CELL SURFACE, G PROTEIN COUPLED RECEPTOR |
552 | Gene ID |
AVPR V1a | dGene Synonym |
AVPR1 | dGene Synonym |
G PROTEIN COUPLED RECEPTOR |