DGIdb - QUINPIROLE Drug Record

QUINPIROLE chembl:CHEMBL240773

Alternate Names:

QUINPIROLE

Drug Info:

(0 More Sources)

Publications:

Vangveravong S et al., 2011, Synthesis and characterization of selective dopamine D₂ receptor ligands using aripiprazole as the lead compound., Bioorg Med Chem
Kühhorn J et al., 2011, Development of a bivalent dopamine D₂ receptor agonist., J Med Chem
Matera C et al., 2015, Bifunctional compounds targeting both D2 and non-α7 nACh receptors: design, synthesis and pharmacological characterization., Eur J Med Chem
Molero A et al., 2015, A solid-phase combinatorial approach for indoloquinolizidine-peptides with high affinity at D(1) and D(2) dopamine receptors., Eur J Med Chem
Tschammer N et al., 2011, Highly potent 5-aminotetrahydropyrazolopyridines: enantioselective dopamine D3 receptor binding, functional selectivity, and analysis of receptor-ligand interactions., J Med Chem

QUINPIROLE DRD2

Interaction Score: 0.45

Interaction Types & Directionality:

agonist (activating)

Interaction Info:

PMIDs:
21999579 26164842 21536445 25969169 21388142

Sources:
DTC
QUINPIROLE DRD3

Interaction Score: 0.38

Interaction Types & Directionality:

agonist (activating)

Interaction Info:

PMIDs:
21536445

Sources:
DTC
QUINPIROLE TDP1

Interaction Score: 0.2

Interaction Types & Directionality:

n/a

Interaction Info:

PMIDs:
None found

Sources:
DTC
QUINPIROLE THRB

Interaction Score: 0.13

Interaction Types & Directionality:

n/a

Interaction Info:

PMIDs:
None found

Sources:
DTC
QUINPIROLE EHMT2

Interaction Score: 0.01

Interaction Types & Directionality:

n/a

Interaction Info:

PMIDs:
None found

Sources:
DTC

DTC: QUINPIROLE

Version: 02-September-2020

Alternate Names:

CHEMBL240773 ChEMBL Drug ID

Drug Info:

Publications:

Vangveravong S et al., 2011, Synthesis and characterization of selective dopamine D₂ receptor ligands using aripiprazole as the lead compound., Bioorg Med Chem

Tschammer N et al., 2011, Highly potent 5-aminotetrahydropyrazolopyridines: enantioselective dopamine D3 receptor binding, functional selectivity, and analysis of receptor-ligand interactions., J Med Chem

Matera C et al., 2015, Bifunctional compounds targeting both D2 and non-α7 nACh receptors: design, synthesis and pharmacological characterization., Eur J Med Chem

ChemblDrugs: chembl:CHEMBL240773
- Version: ChEMBL_27
Alternate Names:

Drug Info:

Publications:

QUINPIROLE Drug Record

QUINPIROLE chembl:CHEMBL240773

Alternate Names:

Drug Info:

Publications:

QUINPIROLE DRD2

Interaction Types & Directionality:

agonist (activating)

Interaction Info:

PMIDs:
21999579 26164842 21536445 25969169 21388142

Sources:
DTC

QUINPIROLE DRD3

Interaction Types & Directionality:

agonist (activating)

Interaction Info:

PMIDs:
21536445

Sources:
DTC

QUINPIROLE TDP1

Interaction Types & Directionality:

n/a

Interaction Info:

PMIDs:
None found

Sources:
DTC

QUINPIROLE THRB

Interaction Types & Directionality:

n/a

Interaction Info:

PMIDs:
None found

Sources:
DTC

QUINPIROLE EHMT2

Interaction Types & Directionality:

n/a

Interaction Info:

PMIDs:
None found

Sources:
DTC

DTC: QUINPIROLE

Alternate Names:

CHEMBL240773 ChEMBL Drug ID

Drug Info:

ChemblDrugs: chembl:CHEMBL240773

Alternate Names:

Drug Info:

Publications:

QUINPIROLE Drug Record

QUINPIROLE chembl:CHEMBL240773

Alternate Names:

Drug Info:

Publications:

QUINPIROLE DRD2

Interaction Types & Directionality: agonist (activating)

Interaction Info:

PMIDs: 21999579 26164842 21536445 25969169 21388142

Sources: DTC

QUINPIROLE DRD3

Interaction Types & Directionality: agonist (activating)

Interaction Info:

PMIDs: 21536445

Sources: DTC

QUINPIROLE TDP1

Interaction Types & Directionality: n/a

Interaction Info:

PMIDs: None found

Sources: DTC

QUINPIROLE THRB

Interaction Types & Directionality: n/a

Interaction Info:

PMIDs: None found

Sources: DTC

QUINPIROLE EHMT2

Interaction Types & Directionality: n/a

Interaction Info:

PMIDs: None found

Sources: DTC

DTC: QUINPIROLE

Alternate Names: CHEMBL240773 ChEMBL Drug ID

Drug Info:

ChemblDrugs: chembl:CHEMBL240773

Alternate Names:

Drug Info:

Publications:

Interaction Types & Directionality:

agonist (activating)

PMIDs:
21999579 26164842 21536445 25969169 21388142

Sources:
DTC

Interaction Types & Directionality:

agonist (activating)

PMIDs:
21536445

Sources:
DTC

Interaction Types & Directionality:

n/a

PMIDs:
None found

Sources:
DTC

Interaction Types & Directionality:

n/a

PMIDs:
None found

Sources:
DTC

Interaction Types & Directionality:

n/a

PMIDs:
None found

Sources:
DTC

Alternate Names:

CHEMBL240773 ChEMBL Drug ID