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INTEPIRDINE Drug Record

  • Summary
  • Interactions
  • Claims
  • INTEPIRDINE chembl:CHEMBL1083390

    Alternate Names:

    GSK-742457
    GSK742457
    RVT-101
    SB-742457
    INTEPIRDINE

    Drug Info:

    (0 More Sources)

    Publications:

    Krogsgaard-Larsen N et al., 2014, Novel aza-analogous ergoline derived scaffolds as potent serotonin 5-HT₆ and dopamine D₂ receptor ligands., J Med Chem
    Ramírez MJ, 2013, 5-HT6 receptors and Alzheimer's disease., Alzheimers Res Ther
  • INTEPIRDINE   HTR6

    Interaction Score: 28.1

    Interaction Types & Directionality:
    antagonist (inhibitory)

    Interaction Info:
    Mechanism of Interaction Serotonin 6 (5-HT6) receptor antagonist
    Direct Interaction yes

    PMIDs:
    24878269 23607787


    Sources:
    DTC ChemblInteractions TTD

  • DTC: SB-742457

    • Version: 02-September-2020

    Alternate Names:
    CHEMBL1083390 ChEMBL Drug ID

    Drug Info:

    Publications:
    Krogsgaard-Larsen N et al., 2014, Novel aza-analogous ergoline derived scaffolds as potent serotonin 5-HT₆ and dopamine D₂ receptor ligands., J Med Chem

  • TTD: SB-742457

    • Version: 2020.06.01

    Alternate Names:
    D0R9HI TTD Drug ID

    Drug Info:

    Publications:
    Ramírez MJ, 2013, 5-HT6 receptors and Alzheimer's disease., Alzheimers Res Ther

  • ChemblInteractions: CHEMBL1083390

    • Version: chembl_23

    Alternate Names:

    Drug Info:

    Publications:

  • ChemblDrugs: chembl:CHEMBL1083390

    • Version: ChEMBL_27

    Alternate Names:

    Drug Info:

    Publications:

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A finding of a drug-gene interaction or potentially druggable category does not necessarily indicate effectiveness (or lack thereof) of any drug or treatment regimen. A finding of no interaction or no potentially druggable category does not necessarily indicate lack of effectiveness of any drug or treatment regimen. Drug-gene interactions or potentially druggable categories are not presented in ranked order of potential or predicted efficacy.

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DGIdb (v4.2.0 - sha1 afd9f30b) • Last updated 2020-10-21