DGIdb - ELACRIDAR Drug Record

ELACRIDAR chembl:CHEMBL396298

Alternate Names:

ELACRIDAR

Drug Info:

Drug Categories	benzocycloheptenes
Drug Categories	drug resistance, multiple
Drug Categories	heterocyclic compounds, fused-ring
Drug Categories	p-glycoprotein inhibitors

(0 More Sources)

Publications:

Hubensack et al., 2008, Effect of the ABCB1 modulators elacridar and tariquidar on the distribution of paclitaxel in nude mice., J. Cancer Res. Clin. Oncol.
Xiao G et al., 2012, Cerebrospinal fluid can be used as a surrogate to assess brain exposures of breast cancer resistance protein and P-glycoprotein substrates., Drug Metab Dispos

ELACRIDAR ABCG2

Interaction Score: 1.33

Interaction Types & Directionality:

n/a

Interaction Info:

PMIDs:
22266779

Sources:
DTC PharmGKB
ELACRIDAR ABCB1

Interaction Score: 0.34

Interaction Types & Directionality:

n/a

Interaction Info:

PMIDs:
17932689

Sources:
DrugBank PharmGKB

DrugBank: DB04881
- Version: 5.1.7
Alternate Names:

ELACRIDAR DrugBank Drug Name

143664-11-3 CAS Number

CHEMBL396298 ChEMBL ID

Drug Info:

Drug Type small molecule

Drug Groups investigational

Drug Categories bcrp/abcg2 inhibitors

Publications:

Hubensack et al., 2008, Effect of the ABCB1 modulators elacridar and tariquidar on the distribution of paclitaxel in nude mice., J. Cancer Res. Clin. Oncol.
DTC: ELACRIDAR
- Version: 02-September-2020
Alternate Names:

CHEMBL396298 ChEMBL Drug ID

Drug Info:

Publications:

Xiao G et al., 2012, Cerebrospinal fluid can be used as a surrogate to assess brain exposures of breast cancer resistance protein and P-glycoprotein substrates., Drug Metab Dispos
ChemblDrugs: chembl:CHEMBL396298
- Version: ChEMBL_27
Alternate Names:

Drug Info:

Publications:
PharmGKB: elacridar
- Version: 18-August-2020
Alternate Names:

Drug Info:

Publications:

ELACRIDAR	DrugBank Drug Name
143664-11-3	CAS Number
CHEMBL396298	ChEMBL ID

Drug Type	small molecule
Drug Groups	investigational
Drug Categories	bcrp/abcg2 inhibitors

ELACRIDAR Drug Record

ELACRIDAR chembl:CHEMBL396298

Alternate Names:

Drug Info:

Publications:

ELACRIDAR ABCG2

Interaction Types & Directionality: n/a

Interaction Info:

PMIDs: 22266779

Sources: DTC PharmGKB

ELACRIDAR ABCB1

Interaction Types & Directionality: n/a

Interaction Info:

PMIDs: 17932689

Sources: DrugBank PharmGKB

DrugBank: DB04881

Alternate Names: ELACRIDAR DrugBank Drug Name 143664-11-3 CAS Number CHEMBL396298 ChEMBL ID

Drug Info: Drug Type small molecule Drug Groups investigational Drug Categories bcrp/abcg2 inhibitors

Publications: Hubensack et al., 2008, Effect of the ABCB1 modulators elacridar and tariquidar on the distribution of paclitaxel in nude mice., J. Cancer Res. Clin. Oncol.

DTC: ELACRIDAR

Alternate Names: CHEMBL396298 ChEMBL Drug ID

Drug Info:

Publications: Xiao G et al., 2012, Cerebrospinal fluid can be used as a surrogate to assess brain exposures of breast cancer resistance protein and P-glycoprotein substrates., Drug Metab Dispos

ChemblDrugs: chembl:CHEMBL396298

Alternate Names:

Drug Info:

Publications:

PharmGKB: elacridar

Alternate Names:

Drug Info:

Publications:

Interaction Types & Directionality:

n/a

PMIDs:
22266779

Sources:
DTC PharmGKB

Interaction Types & Directionality:

n/a

PMIDs:
17932689

Sources:
DrugBank PharmGKB

Alternate Names:

ELACRIDAR DrugBank Drug Name

143664-11-3 CAS Number

CHEMBL396298 ChEMBL ID

Drug Info:

Drug Type small molecule

Drug Groups investigational

Drug Categories bcrp/abcg2 inhibitors

Publications:

Hubensack et al., 2008, Effect of the ABCB1 modulators elacridar and tariquidar on the distribution of paclitaxel in nude mice., J. Cancer Res. Clin. Oncol.

Alternate Names:

CHEMBL396298 ChEMBL Drug ID

Publications:

Xiao G et al., 2012, Cerebrospinal fluid can be used as a surrogate to assess brain exposures of breast cancer resistance protein and P-glycoprotein substrates., Drug Metab Dispos