DIAZEPAM Drug Record
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DIAZEPAM chembl:CHEMBL12 Approved
Alternate Names:
ALUPRAM 5 ALUPRAM 2 DIALAR FTE DIASTAT RELANIUM VALIUM SOLIS LA-III E-PAM DIAZEPAM INTENSOL RO-5-2807 RO-52807 STESOLID SERENACK TRANIMUL DIZAC Q-PAM PAXEL VALRELEASE DIASTAT ACUDIAL APOZEPAM VIVOL ATENSINE WY-3467 NSC-77518 DIAZEPAM CIV TENSIUM DIAZEPAM ALUPRAM 10 SCRIPTOPAM NSC-169897 DIALAR VALCLAIR METHYL DIAZEPINONE VALIUM® DIASTAT® 7-CHLORO-1,3-DIHYDRO-1-METHYL-5-PHENYL-2H-1,4-BENZODIAZEPIN-2-ONE rxcui:3322 chembl:CHEMBL12 drugbank:00829 chemidplus:439-14-5 pubchem.compound:3016 Drug Info:
Drug Class hypnotics and sedatives Year of Approval 1963 Drug Class Small Molecule Drug Indications anticonvulsant FDA Approval approved Publications:
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Interaction Types & Directionality:
potentiator Interaction Info:
Trial Name diazepam rectal gel Novel drug target Established target Trial Name NRL-01 -
Interaction Types & Directionality:
potentiator Interaction Info:
Trial Name diazepam rectal gel Novel drug target Established target Trial Name NRL-01 -
Interaction Types & Directionality:
potentiator Interaction Info:
Trial Name diazepam rectal gel Novel drug target Established target Trial Name NRL-01 -
Interaction Types & Directionality:
ligand positive modulator (activating) allosteric modulator potentiator Interaction Info:
Direct Interaction? True Endogenous Drug? False Specific Action of the Ligand Positive -
Interaction Types & Directionality:
positive modulator (activating) potentiator Interaction Info:
Mechanism of Interaction GABA-A receptor; anion channel positive allosteric modulator Direct Interaction yes Trial Name diazepam rectal gel -
Interaction Types & Directionality:
positive modulator (activating) allosteric modulator potentiator Interaction Info:
Specific Binding Site for Interaction benzodiazepine site Details of the Assay for Interaction Assay using recombinant GABA<sub>A</sub> channels with subunit composition; α3β1γ2. Specific Action of the Ligand Positive
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Interaction Types & Directionality:
positive modulator (activating) allosteric modulator potentiator Interaction Info:
Direct Interaction yes Mechanism of Interaction GABA-A receptor; anion channel positive allosteric modulator Trial Name diazepam rectal gel
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Interaction Types & Directionality:
positive modulator (activating) potentiator Interaction Info:
Mechanism of Interaction GABA-A receptor; anion channel positive allosteric modulator Direct Interaction yes Trial Name diazepam rectal gel -
Interaction Types & Directionality:
positive modulator (activating) potentiator Interaction Info:
Trial Name diazepam rectal gel Novel drug target Established target Trial Name NRL-01 -
Interaction Types & Directionality:
positive modulator (activating) potentiator Interaction Info:
Direct Interaction yes Mechanism of Interaction GABA-A receptor; anion channel positive allosteric modulator Trial Name diazepam rectal gel -
Interaction Types & Directionality:
positive modulator (activating) potentiator Interaction Info:
Trial Name diazepam rectal gel Novel drug target Established target Trial Name NRL-01 -
Interaction Types & Directionality:
positive modulator (activating) potentiator Interaction Info:
Direct Interaction yes Mechanism of Interaction GABA-A receptor; anion channel positive allosteric modulator Trial Name NRL-01 -
Interaction Types & Directionality:
positive modulator (activating) potentiator Interaction Info:
Direct Interaction yes Mechanism of Interaction GABA-A receptor; anion channel positive allosteric modulator Trial Name diazepam rectal gel -
Interaction Types & Directionality:
positive modulator (activating) potentiator Interaction Info:
Trial Name diazepam rectal gel Novel drug target Established target Trial Name NRL-01 -
Interaction Types & Directionality:
positive modulator (activating) potentiator Interaction Info:
Mechanism of Interaction GABA-A receptor; anion channel positive allosteric modulator Direct Interaction yes Trial Name diazepam rectal gel -
Interaction Types & Directionality:
positive modulator (activating) potentiator Interaction Info:
Trial Name NRL-01 Novel drug target Established target Trial Name diazepam rectal gel -
Interaction Types & Directionality:
positive modulator (activating) potentiator Interaction Info:
Mechanism of Interaction GABA-A receptor; anion channel positive allosteric modulator Direct Interaction yes -
Interaction Types & Directionality:
positive modulator (activating) Interaction Info:
Mechanism of Interaction GABA-A receptor; anion channel positive allosteric modulator Direct Interaction yes -
Interaction Types & Directionality:
positive modulator (activating) Interaction Info:
Mechanism of Interaction GABA-A receptor; anion channel positive allosteric modulator Direct Interaction yes
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Alternate Names:
DIAZEPAM Primary Drug Name Drug Info:
Year of Approval 1963 Drug Class hypnotics and sedatives Publications:
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- Version: January-2014
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Drug Info:
FDA Approval approved Drug Indications anticonvulsant Drug Class Small Molecule Publications:
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Alternate Names:
C28982 NCI drug code Drug Info:
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Alternate Names:
CHEMBL12 ChEMBL Drug ID Drug Info:
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Drug Info:
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D07JVL TTD Drug ID Drug Info:
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- Version: 29-September-2020
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DIAZEPAM GuideToPharmacology Ligand Name Drug Info:
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- Version: ChEMBL_27
Alternate Names:
Drug Info:
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- Version: chembl_23
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Drug Info:
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Alternate Names:
Drug Info:
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