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CHEMBL1077391 Drug Record

  • Summary
  • Interactions
  • Claims
  • CHEMBL1077391 chembl:CHEMBL1077391

    Alternate Names:

    RO-4882224

    Drug Info:

    (0 More Sources)

    Publications:

    Knust H et al., 2009, The discovery and unique pharmacological profile of RO4938581 and RO4882224 as potent and selective GABAA alpha5 inverse agonists for the treatment of cognitive dysfunction., Bioorg Med Chem Lett
  • CHEMBL1077391   GABRB3

    Interaction Score: 0.66

    Interaction Types & Directionality:
    n/a

    Interaction Info:

    PMIDs:
    19762240


    Sources:
    DTC

  • CHEMBL1077391   GABRG2

    Interaction Score: 0.62

    Interaction Types & Directionality:
    n/a

    Interaction Info:

    PMIDs:
    19762240


    Sources:
    DTC

  • CHEMBL1077391   GABRA5

    Interaction Score: 0.56

    Interaction Types & Directionality:
    n/a

    Interaction Info:

    PMIDs:
    19762240


    Sources:
    DTC

  • DTC: RO-4882224

    • Version: 02-September-2020

    Alternate Names:
    CHEMBL1077391 ChEMBL Drug ID

    Drug Info:

    Publications:
    Knust H et al., 2009, The discovery and unique pharmacological profile of RO4938581 and RO4882224 as potent and selective GABAA alpha5 inverse agonists for the treatment of cognitive dysfunction., Bioorg Med Chem Lett

  • ChemblDrugs: chembl:CHEMBL1077391

    • Version: ChEMBL_27

    Alternate Names:

    Drug Info:

    Publications:

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DGIdb (v4.2.0 - sha1 afd9f30b) • Last updated 2020-10-21