ASENAPINE Drug Record
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ASENAPINE chembl:CHEMBL3187365 Approved
Alternate Names:
ASENAPINE SYCREST Drug Info:
Drug Class antipsychotic agents Year of Approval 2009 FDA Approval approved Drug Class Small molecule Drug Indications antipsychotic agent Drug Categories acid reducers Drug Categories adrenergic alpha-1 receptor antagonists Drug Categories adrenergic alpha-antagonists Drug Categories adrenergic antagonists Drug Categories agents that produce hypertension Drug Categories antidepressive agents Drug Categories cytochrome p-450 cyp2d6 inhibitors (weak) Drug Categories cytochrome p-450 cyp2d6 substrates Drug Categories cytochrome p-450 cyp3a substrates Drug Categories cytochrome p-450 enzyme inhibitors Drug Categories cytochrome p-450 substrates Drug Categories dopamine antagonists Drug Categories dopamine d2 receptor antagonists Drug Categories heterocyclic compounds, fused-ring Drug Categories histamine antagonists Drug Categories histamine h1 antagonists Drug Categories histamine h2 antagonists Drug Categories neurotoxic agents Drug Categories qtc prolonging agents Drug Categories serotonergic drugs shown to increase risk of serotonin syndrome Drug Categories serotonin agents Drug Categories serotonin receptor agonists Drug Categories ugt1a4 substrates Publications:
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Interaction Types & Directionality:
antagonist (inhibitory) Interaction Info:
Trial Name Asenapine Novel drug target Established target -
Interaction Types & Directionality:
antagonist (inhibitory) Interaction Info:
Novel drug target Established target Trial Name Asenapine -
Interaction Types & Directionality:
antagonist (inhibitory) Interaction Info:
Novel drug target Established target Trial Name Asenapine -
Interaction Types & Directionality:
antagonist (inhibitory) Interaction Info:
Trial Name Asenapine Novel drug target Established target -
Interaction Types & Directionality:
agonist (activating) antagonist (inhibitory) Interaction Info:
Endogenous Drug? False Specific Action of the Ligand Full agonist Trial Name Asenapine -
Interaction Types & Directionality:
antagonist (inhibitory) Interaction Info:
Trial Name Asenapine Novel drug target Established target -
Interaction Types & Directionality:
antagonist (inhibitory) Interaction Info:
Trial Name Asenapine Novel drug target Established target -
Interaction Types & Directionality:
antagonist (inhibitory) Interaction Info:
Novel drug target Established target Trial Name Asenapine -
Interaction Types & Directionality:
antagonist (inhibitory) Interaction Info:
Trial Name Asenapine Novel drug target Established target -
Interaction Types & Directionality:
antagonist (inhibitory) Interaction Info:
Trial Name Asenapine Novel drug target Established target Direct Interaction? True -
Interaction Types & Directionality:
agonist (activating) antagonist (inhibitory) Interaction Info:
Novel drug target Established target Trial Name Asenapine Endogenous Drug? False -
Interaction Types & Directionality:
antagonist (inhibitory) Interaction Info:
Novel drug target Established target Trial Name Asenapine -
Interaction Types & Directionality:
antagonist (inhibitory) Interaction Info:
Trial Name Asenapine Novel drug target Established target Specific Action of the Ligand Antagonist -
Interaction Types & Directionality:
agonist (activating) Interaction Info:
Specific Action of the Ligand Full agonist Endogenous Drug? False -
Interaction Types & Directionality:
antagonist (inhibitory) Interaction Info:
Trial Name Asenapine Novel drug target Established target -
Interaction Types & Directionality:
antagonist (inhibitory) Interaction Info:
Specific Action of the Ligand Antagonist Endogenous Drug? False Trial Name Asenapine -
Interaction Types & Directionality:
antagonist (inhibitory) Interaction Info:
Trial Name Asenapine Novel drug target Established target -
Interaction Types & Directionality:
antagonist (inhibitory) Interaction Info:
Trial Name Asenapine Novel drug target Established target -
Interaction Types & Directionality:
antagonist (inhibitory) Interaction Info:
Trial Name Asenapine Novel drug target Established target -
Interaction Types & Directionality:
agonist (activating) Interaction Info:
Specific Action of the Ligand Full agonist Endogenous Drug? False
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Alternate Names:
65576-45-6 CAS Number Saphris Drug Brand Secuado Drug Brand Drug Info:
Drug Type small molecule Drug Groups approved Drug Categories acid reducers Publications:
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- Version: January-2014
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Drug Info:
Drug Indications antipsychotic agent Drug Class Small molecule FDA Approval approved Publications:
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Drug Info:
Year of Approval 2009 Drug Class antipsychotic agents Publications:
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D00JRA TTD Drug ID Drug Info:
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- Version: ChEMBL_27
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Drug Info:
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- Version: 29-September-2020
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Drug Info:
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