5467 |
PEROXISOME PROLIFERATOR ACTIVATED RECEPTOR DELTA |
PPARD |
FAAR |
NR1C2 |
NUC1 |
NUCI |
NUCII |
PPARB |
600409 |
9235 |
ENSG00000112033 |
OTTHUMG00000014567 |
PEROXISOME PROLIFERATOR ACTIVATED RECEPTOR DELTA (PPAR-DELTA) (PPAR- BETA) (NUCLEAR HORMONE RECEPTOR 1) (NUC1) (NUCI). [SOURCE:UNIPROT/SWISSPROT;ACC:Q03181] |
BE0001007 |
Q03181 |
PA33557 |
peroxisome proliferator-activated receptor delta |
PPAR-beta |
Nuclear hormone receptor 1 |
Nuclear receptor subfamily 1 group C member 2 |
Peroxisome proliferator-activated receptor beta |
PPAR-delta |
PPARD_HUMAN |
TTDC00069 |
PPARDELTA |
PEROXISOME PROLIFERATOR ACTIVATED RECEPTOR BETA/DELTA |
594 |
Peroxisome proliferator-activated receptor-β/δ |
NP_006229 |
NM_177435 |
Human Readable Name | DRUGGABLE GENOME |
Initial Gene Query | NR1C2 |
Counted Citations from 1950-2000 | 900 |
Gene Category | Nuclear Hormone Receptors |
Is VIP | false |
Has Variant Annotation | true |
Human Readable Name | NUCLEAR HORMONE RECEPTOR |
Target Class | Receptors |
Target Subclass | Nuclear receptor |
Gene Biotype | PROTEIN_CODING" |
Interpro Acc | IPR000536 |
Interpro Name | Nuclear hormone receptor, ligand-binding, core |
Uniprot Status | Swiss-Prot |
Interpro Type | Domain |
Uniprot Evidence | 1: Evidence at protein level |
Interpro Short Name | Nucl_hrmn_rcpt_lig-bd_core |
GuideToPharmacology Gene Category Name | 1C. Peroxisome proliferator-activated receptors |
GuideToPharmacology Gene Category ID | 86 |
GuideToPharmacology Gene Type | nhr |
agonist |
Specific Action of the Ligand | Full agonist |
Endogenous Drug? | False |
Direct Interaction? | False |
agonist |
Trial Name | DB-959 |
Novel drug target | Established target |
Mechanism of Interaction | Peroxisome proliferator-activated receptor delta agonist |
agonist |
Trial Name | KD3010 |
Novel drug target | Established target |
Mechanism of Interaction | Peroxisome proliferator-activated receptor delta agonist |
agonist |
Specific Action of the Ligand | Full agonist |
Endogenous Drug? | False |
agonist |
Specific Action of the Ligand | Full agonist |
Endogenous Drug? | False |
Direct Interaction? | False |
agonist |
Specific Action of the Ligand | Full agonist |
Endogenous Drug? | False |
Direct Interaction? | False |
agonist |
Specific Action of the Ligand | Full agonist |
Endogenous Drug? | False |
agonist |
Specific Action of the Ligand | Full agonist |
Endogenous Drug? | False |
agonist |
Specific Action of the Ligand | Full agonist |
Endogenous Drug? | False |
agonist |
Specific Action of the Ligand | Full agonist |
Endogenous Drug? | True |
Direct Interaction? | False |
antagonist |
Specific Action of the Ligand | Antagonist |
Endogenous Drug? | False |
agonist |
Trial Name | CER-002 |
Novel drug target | Established target |
Mechanism of Interaction | Peroxisome proliferator-activated receptor delta agonist |
agonist |
Trial Name | MBX-8025 |
Novel drug target | Established target |
Mechanism of Interaction | Peroxisome proliferator-activated receptor delta agonist |
agonist |
Mechanism of Interaction | Peroxisome proliferator-activated receptor agonist |
Direct Interaction | yes |
agonist |
Mechanism of Interaction | Peroxisome proliferator-activated receptor delta agonist |
Direct Interaction | yes |
agonist |
agonist |
negative modulator |
agonist |
agonist |
Mechanism of Interaction | Peroxisome proliferator-activated receptor agonist |
Direct Interaction | yes |
agonist |
agonist |
n/a |
Trial Name | AMR102 |
Novel drug target | Established target |
n/a |
n/a |
n/a |
n/a |
n/a |
n/a |
n/a |
n/a |
PPARD | Ensembl Gene Name |
Gene Biotype | PROTEIN_CODING" |
PPARD | Display Id |
PEROXISOME PROLIFERATOR ACTIVATED RECEPTOR DELTA (PPAR-DELTA) (PPAR- BETA) (NUCLEAR HORMONE RECEPTOR 1) (NUC1) (NUCI). [SOURCE:UNIPROT/SWISSPROT;ACC:Q03181] | Description |
ENSG00000112033 | Ensembl Gene Id |
Human Readable Name | DRUGGABLE GENOME |
peroxisome proliferator-activated receptor delta | Gene Name |
ENSG00000112033 | Ensembl Gene Id |
5467 | Entrez Gene Id |
Is VIP | false |
Has Variant Annotation | true |
PPARD | Gene Symbol |
5467 | Entrez Gene Id |
Human Readable Name | NUCLEAR HORMONE RECEPTOR |
5467 | Entrez Gene ID |
Initial Gene Query | NR1C2 |
Counted Citations from 1950-2000 | 900 |
Gene Category | Nuclear Hormone Receptors |
5467 | Entrez Gene Id |
PPARD_HUMAN | Uniprot Id |
ENSG00000112033 | Ensembl Gene Id |
Interpro Acc | IPR000536 |
Human Readable Name | NUCLEAR HORMONE RECEPTOR |
Interpro Name | Nuclear hormone receptor, ligand-binding, core |
peroxisome proliferator-activated receptor delta | HUGO Gene Name |
9235 | HUGO Gene ID |
PPARD | Gene Symbol |
GuideToPharmacology Gene Category Name | 1C. Peroxisome proliferator-activated receptors |
GuideToPharmacology Gene Category ID | 86 |
GuideToPharmacology Gene Type | nhr |
PPARD | Gene Symbol |
Target Class | Receptors |
Target Subclass | Nuclear receptor |
PPARD | DrugBank Gene Name |
Q03181 | UniProt Accession |
5467 | Entrez Gene Id |
Peroxisome proliferator-activated receptor-β/δ | GuideToPharmacology Name |
Q03181 | UniProtKB ID |
5467 | Entrez Gene Id |
PPAR-BETA | Gene Synonym |
NUCLEAR HORMONE RECEPTOR 1 | Gene Synonym |
ENSG00000112033 | Gene Symbol |
PPARD | Ensembl Id |
Q03181 | UniProtKB ID |
PPARD_HUMAN | GO Gene Synonym |
NR1C2 | GO Gene Synonym |
PPARB | GENE_SYMBOL |
PPARD | GENE_SYMBOL |
Peroxisome proliferator-activated receptor delta | UNIPROT |